Pyrazinyl-substituted aminoazoles as covalent inhibitors of thrombin: synthesis, structure, and anticoagulant properties.

Imberg, L.; Siutkina, A. I.; Erbacher, C.; Schmidt, J.; Broekmans, D. F.; Ovsepyan, R. A.; Daniliuc, C. G.; de Oliveira, E. G.; Serafim, M. S. M.; O´Donoghue, A.; Pillaiyar, T.; Panteleev, M., A.; Poso, A.; Kalinina, S.; Bermudez M.; Nekipelov, K.; Bendas G.; Karst, U.; Kalinin, D. V.

Research article (journal) | Peer reviewed

Details about the publication

JournalACS Pharmacology & Translational Science
Volume8
Issue1
StatusPublished
Release year2024
DOI10.1021/acsptsci.4c00515
KeywordsAnticoagulants, Thrombosis, Thrombin

Authors from the University of Münster

Kalinin, Dmitrii
Independent Junior Research Group Dmitrii Kalinin
Kalinina, Svetlana
Independent Junior Research Group Svetlana Kalinina