Radical Reactions of Alkyl 2-Bromo-2,2-difluoroacetates with Vinyl Ethers: “Omitted” Examples and Application for the Synthesis of 3,3-Difluoro-GABA

Kondratov IS, Bugera MY, Tolmachova NA, Posternak GG, Daniliuk CG, Haufe G (2015)
In: Journal of Organic Chemistry, 80
Type of Publication: Research article (journal)

Synthesis and Physical-chemical Properties of 3-Fluorocyclobutyl Amines

Chernykh AX, Radchenko DX, Kondratov IS, Tolmachova NA, Datsenko OX, Kurkunov MA, Zozulya SX, Kheylik YX, Bartels K, Daniliuk CG, Haufe G (2015)
In: European Journal of Organic Chemistry, 2015
Type of Publication: Research article (journal)

Synthesis of new fluorinated analogs of GABA, Pregabalin bioisosteres, and their effects on [H-3]GABA uptake by rat brain nerve terminals

Borisova T, Pozdnyakova N, Shaitanova E, Gerus I, Dudarenko M, Mironets R, Haufe G, Kukhar V (2015)
In: Bioorganic & Medicinal Chemistry, 23
Type of Publication: Research article (journal)

New Matrix-Metallo-Proteinase Inhibitors Based on γ-Fluorinated α-aminocarboxylic and α-aminohydroxamic acids

Behrends M, Wagner S, Kopka K, Schröer S, Schober O, Schäfers M, Kumbhar S, Waller M, Haufe G (2015)
In: Bioorganic & Medicinal Chemistry, 23
Type of Publication: Research article (journal)

Sphingosin-1-phosphate receptor 3 promotes leukocyte rolling by mobilizing endothelial P-selectin

Nussbaum C, Bannenberg S, Keul P, Gräler MH, Goncalves-De-Albuquerque CF, Korhonen H, von Wnuk Lipinski K, Heusch G, Neto HCF, Rohwedder I, Göthert J, Prasad VP, Haufe G, Lange-Sperandio B, Offermanns S, Sperandio M, Levkau B (2015)
In: Nature Communications, 7416
Type of Publication: Research article (journal)

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Radical Reactions of Alkyl 2-Bromo-2,2-difluoroacetates with Vinyl Ethers: “Omitted” Examples and Application for the Synthesis of 3,3-Difluoro-GABA Kondratov IS, Bugera MY, Tolmachova NA, Posternak GG, Daniliuk CG, Haufe G (2015) In: Journal of Organic Chemistry, 80 Type of Publication: Research article (journal)
New Fluorinated Agonists for Targeting the Sphingosin-1-Phosphate Receptor 1 (S1P1) Shaikh RS, Keul P, Schäfers M, Levkau B, Haufe G (2015) In: Bioorganic & Medicinal Chemistry Letters, 25 Type of Publication: Research article (journal)
Synthesis and Physical-chemical Properties of 3-Fluorocyclobutyl Amines Chernykh AX, Radchenko DX, Kondratov IS, Tolmachova NA, Datsenko OX, Kurkunov MA, Zozulya SX, Kheylik YX, Bartels K, Daniliuk CG, Haufe G (2015) In: European Journal of Organic Chemistry, 2015 Type of Publication: Research article (journal)
Novel fluorine-18 labeled 5-(1-pyrrolidinylsulfonyl)-7-azaisatin derivatives as potential PET tracers for in vivo imaging of activated caspases in apoptosis Waldmann CM, Hermann S, Faust A, Riemann R, Schober O, Schäfers M, Haufe G, Kopka K (2015) In: Bioorganic & Medicinal Chemistry, 23 Type of Publication: Research article (journal)
Synthesis of new fluorinated analogs of GABA, Pregabalin bioisosteres, and their effects on [H-3]GABA uptake by rat brain nerve terminals Borisova T, Pozdnyakova N, Shaitanova E, Gerus I, Dudarenko M, Mironets R, Haufe G, Kukhar V (2015) In: Bioorganic & Medicinal Chemistry, 23 Type of Publication: Research article (journal)
Studies of Genotoxicity and Mutagenicity of Nitroimidazoles: Demystifying this Critical Relationship with the Nitro Group Boechat N, Carvalho AS, Bastos MM, Salomão K, De Castro SL, Araujo-Lima CF, Mello FVC, Felzenszwalb I, Aiub C, Condre TR, Zamith HPS, Skupin R, Haufe G (2015) In: Memórias do Instituto Oswaldo Cruz, 110 Type of Publication: Research article (journal)
New Matrix-Metallo-Proteinase Inhibitors Based on γ-Fluorinated α-aminocarboxylic and α-aminohydroxamic acids Behrends M, Wagner S, Kopka K, Schröer S, Schober O, Schäfers M, Kumbhar S, Waller M, Haufe G (2015) In: Bioorganic & Medicinal Chemistry, 23 Type of Publication: Research article (journal)
Synthesis and Evaluation of Fluorinated Fingolimod (FTY720) Analogues for Sphingosine-1-Phosphate Receptor Molecular Imaging by Positron Emission Tomography Shaikh RS, Schilson SS, Wagner S, Hermann S, Keul P, Levkau B, Schäfedrs M, Haufe G (2015) In: Journal of Medicinal Chemistry, 2015 Type of Publication: Research article (journal)
Sphingosin-1-phosphate receptor 3 promotes leukocyte rolling by mobilizing endothelial P-selectin Nussbaum C, Bannenberg S, Keul P, Gräler MH, Goncalves-De-Albuquerque CF, Korhonen H, von Wnuk Lipinski K, Heusch G, Neto HCF, Rohwedder I, Göthert J, Prasad VP, Haufe G, Lange-Sperandio B, Offermanns S, Sperandio M, Levkau B (2015) In: Nature Communications, 7416 Type of Publication: Research article (journal)
Synthesis of New Trifluoromethyl Containing Polysubstituted Aromatic Compounds by Diels-Alder Reaction of Ethyl 3-Benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate Kondratov IS, Tolmachova NA, Dolovanyuk VG, Gerus II, Daniliuk CG, Haufe G (2015) In: European Journal of Organic Chemistry, 2015 Type of Publication: Research article (journal)