Naphtho[1,2-b][1,4]diazepinedione-based P2X4 Receptor Antagonists from Structure-Activity Relationships Studies toward PET Tracer Development

Erlitz, KS; Prinz, AK; Wagner, S; Massa, J; Dunker, C; Höhl, M; Griep, A; McMaus, RM; Schelhaas, S; Koch, O; Junker, A (2025)

In: Journal of Medicinal Chemistry, 68.

Research article (journal)

Synthesis, radiosynthesis and biochemical evaluation of fluorinated analogues of sphingosine-1-phosphate receptor 3 specific antagonists using PET

Puspha Prasad, Vysakh; Wagner, Stefan; Keul, Petra; Hermann, Sven; Levkau, Bodo; Schäfers, Michael; Haufe, Günter (2024)

In: Bioorganic & Medicinal Chemistry, 104, 117697.

Research article (journal)

Translational imaging of the fibroblast activation protein (FAP) using the new ligand [68Ga]Ga-OncoFAP-DOTAGA.

Backhaus P; Gierse F; Burg MC; Büther F; Asmus I; Dorten P; Cufe J; Roll W; Neri D; Cazzamalli S; Millul J; Mock J; Galbiati A; Zana A; Schäfers KP; Hermann S; Weckesser M; Tio J; Wagner S; Breyholz HJ; Schäfers M (2022)

In: European Journal of Nuclear Medicine and Molecular Imaging, 49(6).

Research article (journal)

Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors

Wagner S, de Moura Gatti F, Silva DG, Ortiz Zacarias NV, Zweemer AJM, Hermann S, De Maria M, Koch M, Weiss C, Schepmann D, Heitman LH, Tschammer N, Kopka K, Junker A (2021)

In: ChemMedChem, 16.

Research article (journal)

Initial experience with [18F]DPA-714 TSPO-PET to image inflammation in primary angiitis of the central nervous system

Backhaus P, Roll W, Beuker C, Zinnhardt B, Seifert R, Wenning C, Eisenblätter M, Thomas C, Schmidt-Pogoda A, Strunk D, Wagner S, Faust A, Tüttelmann F, Röpke A, Jacobs AH, Stummer W, Wiendl H, Meuth S, Schäfers M, Grauer O, Minnerup J (2020)

In: European Journal of Nuclear Medicine and Molecular Imaging, 47.

Research article (journal)

Publications

Contact

Top-Links

Synthesis of piperazine-based fluorinated fibroblast activation protein inhibitors for the development of a novel 18F-labeled PET imaging probe. Köchel R; Wagner S; Schwegmann K; Schäfers M; Breyholz HJ; Wünsch B (2025) In: European Journal of Medicinal Chemistry, 290. Research article (journal)
Naphtho[1,2-b][1,4]diazepinedione-based P2X4 Receptor Antagonists from Structure-Activity Relationships Studies toward PET Tracer Development Erlitz, KS; Prinz, AK; Wagner, S; Massa, J; Dunker, C; Höhl, M; Griep, A; McMaus, RM; Schelhaas, S; Koch, O; Junker, A (2025) In: Journal of Medicinal Chemistry, 68. Research article (journal)
Novel [18F]Fluorine-Based PET Tracers with Polar But Nonbasic Linkers to Image the Fibroblast Activation Protein in the Microenvironment of Tumors Köchel, Ricardo; Schwegmann, Katrin; Breyholz, Hans-Jörg; Schäfers, Michael; Wagner, Stefan; Wünsch, Bernhard (2025) In: Journal of Medicinal Chemistry, 68(15). Research article (journal)
Synthesis, radiosynthesis and biochemical evaluation of fluorinated analogues of sphingosine-1-phosphate receptor 3 specific antagonists using PET Puspha Prasad, Vysakh; Wagner, Stefan; Keul, Petra; Hermann, Sven; Levkau, Bodo; Schäfers, Michael; Haufe, Günter (2024) In: Bioorganic & Medicinal Chemistry, 104, 117697. Research article (journal)
Interrogating Glioma-Associated Microglia and Macrophage Dynamics Under CSF-1R Therapy with Multitracer In Vivo PET/MRI Foray, Claudia; Barca, Cristina; Winkeler, Alexander; Wagner, Stefan; Hermann, Sven; Schafers, Michael; grauer, Oliver; Zinnhardt, Bastian; Jacobs, Andreas (2022) In: Journal of Nuclear Medicine, 63(9). Research article (journal)
Translational imaging of the fibroblast activation protein (FAP) using the new ligand [68Ga]Ga-OncoFAP-DOTAGA. Backhaus P; Gierse F; Burg MC; Büther F; Asmus I; Dorten P; Cufe J; Roll W; Neri D; Cazzamalli S; Millul J; Mock J; Galbiati A; Zana A; Schäfers KP; Hermann S; Weckesser M; Tio J; Wagner S; Breyholz HJ; Schäfers M (2022) In: European Journal of Nuclear Medicine and Molecular Imaging, 49(6). Research article (journal)
Imaging TMZ-induced changes in the myeloid glioma microenvironment Foray C, Valtorta S, Barca C, Winkeler A, Roll W, Müther M, Wagner S, Hermann S, Schäfers M, Grauer O, Moresco RM, Zinnhardt B, Jacobs AH (2021) In: Theranostics, 11. Research article (journal)
Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors Wagner S, de Moura Gatti F, Silva DG, Ortiz Zacarias NV, Zweemer AJM, Hermann S, De Maria M, Koch M, Weiss C, Schepmann D, Heitman LH, Tschammer N, Kopka K, Junker A (2021) In: ChemMedChem, 16. Research article (journal)
Do fasting or high caloric drinks affect the physiological uptake of fluorine-18 prostate-specific membrane antigen-1007 in liver and bowel? Rahbar K, Afshar-Oromieh A, Seifert R, Wagner S, Schäfers M, Bögemann M, Weckesser M (2020) In: World Journal of Nuclear Medicine, 19. Research article (journal)
Initial experience with [18F]DPA-714 TSPO-PET to image inflammation in primary angiitis of the central nervous system Backhaus P, Roll W, Beuker C, Zinnhardt B, Seifert R, Wenning C, Eisenblätter M, Thomas C, Schmidt-Pogoda A, Strunk D, Wagner S, Faust A, Tüttelmann F, Röpke A, Jacobs AH, Stummer W, Wiendl H, Meuth S, Schäfers M, Grauer O, Minnerup J (2020) In: European Journal of Nuclear Medicine and Molecular Imaging, 47. Research article (journal)