10-(4-Phenylpiperazine-1-carbonyl)acridin-9(10H)-ones and related compounds: Synthesis, antiproliferative activity and inhibition of tubulin polymerization

Waltemate J., Ivanov I., Ghasemi J. B., Aghaee E., Daniliuc C. G., Müller K., Prinz H. (2021)
In: Bioorganic and Medicinal Chemistry Letters, 32
Type of Publication: Research article (journal)

Synthesis, antiproliferative activity evaluation and 3D-QSAR study of naphthoquinone derivatives as potential anti-colorectal cancer agents

Acuña, J Piermattey, J Caro, D Barrios, L Bannwitz, S López, J Ocampo, Y Vivas-Reyes, R Gaitán, R Aristizábal, F Müller, K Franco, L (2018)
In: Molecules, 23
Type of Publication: Research article (journal)

Oxadiazole-substituted naphtho[2,3-b]thiophene-4,9-diones as potent inhibitors of keratinocyte hyperproliferation. Structure−activity relationships of the tricyclic quinone…

Basoglu A, Dirkmann S, Zahedi Golpayegani N, Vortherms S, Tentrop J, Nowottnik D, Prinz H, Fröhlich R, Müller K (2017)
In: European Journal of Medicinal Chemistry, 134
Type of Publication: Research article (journal)

8-Halo-substituted naphtho[2,3-b]thiophene-4,9-diones as redox-active inhibitors of keratinocyte hyperproliferation with reduced membrane-damaging properties

Lindenschmidt C, Krane D, Vortherms S, Hilbig L, Prinz H, Müller K (2016)
In: European Journal of Medicinal Chemistry, 110
Type of Publication: Research article (journal)

Synthesis and structure–activity relationships of lapacho analogues. 2. Modification of the basic naphtho[2,3-b]furan-4,9-dione, redox activation, and suppression of human…

Bannwitz, V, Krane, D, Vortherms, S, Kalin, T, Lindenschmidt, C, Zahedi Golpayegani, N, Tentrop, J, Prinz, H, Müller, K (2014)
In: Journal of Medicinal Chemistry, 57(14)
Type of Publication: Research article (journal)

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10-(4-Phenylpiperazine-1-carbonyl)acridin-9(10H)-ones and related compounds: Synthesis, antiproliferative activity and inhibition of tubulin polymerization Waltemate J., Ivanov I., Ghasemi J. B., Aghaee E., Daniliuc C. G., Müller K., Prinz H. (2021) In: Bioorganic and Medicinal Chemistry Letters, 32 Type of Publication: Research article (journal)
A promising naphthoquinone [8-hydroxy-2-(2-thienylcarbonyl)naphtho[2,3-b]thiophene-4,9-dione] exerts anti-colorectal cancer activity through ferroptosis and inhibition of MAPK… Caro D, Rivera, D. E., Ocampo Y., Müller K., Franco, L. A. (2020) In: Open Chemistry, 18 Type of Publication: Research article (journal)
Synthesis, antiproliferative activity evaluation and 3D-QSAR study of naphthoquinone derivatives as potential anti-colorectal cancer agents Acuña, J Piermattey, J Caro, D Barrios, L Bannwitz, S López, J Ocampo, Y Vivas-Reyes, R Gaitán, R Aristizábal, F Müller, K Franco, L (2018) In: Molecules, 23 Type of Publication: Research article (journal)
Napabucasin and Related Heterocycle-Fused Naphthoquinones as STAT3 Inhibitors with Antiproliferative Activity against Cancer Cells Löcken H, Clamor C, Müller K (2018) In: Journal of Natural Products, 81(7) Type of Publication: Research article (journal)
Oxadiazole-substituted naphtho[2,3-b]thiophene-4,9-diones as potent inhibitors of keratinocyte hyperproliferation. Structure−activity relationships of the tricyclic quinone… Basoglu A, Dirkmann S, Zahedi Golpayegani N, Vortherms S, Tentrop J, Nowottnik D, Prinz H, Fröhlich R, Müller K (2017) In: European Journal of Medicinal Chemistry, 134 Type of Publication: Research article (journal)
N-Heterocyclic (4-phenylpiperazin-1-yl)methanones derived from phenoxazine and phenothiazine as highly potent inhibitors of tubulin polymerization Prinz H, Ridder A, Vogel K, Böhm KJ, Ivanov I, Ghasemi JB, Aghaee E, Müller K (2017) In: Journal of Medicinal Chemistry, 60(2) Type of Publication: Research article (journal)
8-Halo-substituted naphtho[2,3-b]thiophene-4,9-diones as redox-active inhibitors of keratinocyte hyperproliferation with reduced membrane-damaging properties Lindenschmidt C, Krane D, Vortherms S, Hilbig L, Prinz H, Müller K (2016) In: European Journal of Medicinal Chemistry, 110 Type of Publication: Research article (journal)
Inhibitory effect of phenothiazine- and phenoxazine-derived chloroacetamides on Leishmania major growth and Trypanosoma brucei trypanothione reductase Marcu A, Schurigt U, Müller K, Moll H, Krauth-Siegel RL, Prinz H (2016) In: European Journal of Medicinal Chemistry, 108 Type of Publication: Research article (journal)
Synthesis and structure–activity relationships of lapacho analogues. 2. Modification of the basic naphtho[2,3-b]furan-4,9-dione, redox activation, and suppression of human… Bannwitz, V, Krane, D, Vortherms, S, Kalin, T, Lindenschmidt, C, Zahedi Golpayegani, N, Tentrop, J, Prinz, H, Müller, K (2014) In: Journal of Medicinal Chemistry, 57(14) Type of Publication: Research article (journal)
Synthesis and structure–sctivity relationships of lapacho analogues. 1. Suppression of human keratinocyte hyperproliferation by 2-substituted naphtho[2,3-b]furan-4,9-diones,… Reichstein A, Vortherms S, Bannwitz S, Tentrop J, Prinz H, Müller K (2012) In: Journal of Medicinal Chemistry, 55(16) Type of Publication: Research article (journal)