Di Pizio, A; Bermudez, M; De Graaf, C; Jockers, R (2023)

In: Frontiers in endocrinology, 14, 1189508. doi:10.3389/fendo.2023.1189508

Editorial (journal) | Peer reviewed | Published

Community guidelines for GPCR ligand bias: IUPHAR review 32

Kolb, P; Kenakin, T; Alexander, S; Bermudez, M; Bohn, L; Breinholt; C; Bouvier, M; Hill, S; Kostenis, E; Martemyanov, K; Neubig, R; Onaran, O; Rajagopal, S; Roth, B; Selent, J; Shukla, A; Sommer, M; Gloriam D (2022)

In: British Journal of Pharmacology, 179(14), 3651-3674. doi:10.1111/bph.15811

Review article (journal) | Peer reviewed | Published

Antinociceptive Efficacy of the µ-Opioid/Nociceptin Peptide-Based Hybrid KGNOP1 in Inflammatory Pain without Rewarding Effects in Mice: An Experimental Assessment and Molecular Docking

Dumitrascuta M, Bermudez M, Trovato O, Neve JD, Ballet S, Wolber G, Spetea M (2021)

In: Molecules, 26, 3267-3267. doi:10.3390/molecules26113267

Research article (journal) | Peer reviewed | Published

Biological Characterization, Mechanistic Investigation and Structure‐Activity Relationships of Chemically Stable TLR2 Antagonists

Bermudez M, Grabowski M, Murgueitio MS, Tiemann M, Varga P, Rudolf T, Wolber G, Weindl G, Rademann J (2020)

In: ChemMedChem, 15, 1364-1371. doi:10.1002/cmdc.202000060

Research article (journal) | Peer reviewed | Published

Mechanistic Understanding of Peptide Analogues, DALDA, [Dmt1]DALDA, and KGOP01, Binding to the Mu Opioid Receptor

Dumitrascuta M, Bermudez M, Ballet S, Wolber G, Spetea M (2020)

In: Molecules, 25, 2087. doi:10.3390/molecules25092087

Research article (journal) | Peer reviewed | Published

Structural determinants of sphingosine-1-phosphate receptor selectivity Wunsch, F; Nguyen, TN; Wolber, G; Bermudez, M (2023) In: Archiv der Pharmazie / Chemistry in Life Sciences, 356(12), 2300387. doi:10.1002/ardp.202300387 Research article (journal) \| Peer reviewed \| Published
Peptide-binding GPCRs coming of age Di Pizio, A; Bermudez, M; De Graaf, C; Jockers, R (2023) In: Frontiers in endocrinology, 14, 1189508. doi:10.3389/fendo.2023.1189508 Editorial (journal) \| Peer reviewed \| Published
Hybridization into a Bitopic Ligand Increased Muscarinic Receptor Activation for Isopilocarpine but Not for Pilocarpine Derivatives Heinz, C; Bermudez, M; Jaiswal, N; Große, C; Kauk, M; Hoffmann, C; Holzgrabe, U (2023) In: Journal of Natural Products, 86(4), 869-881. doi:10.1021/acs.jnatprod.2c01079 Research article (journal) \| Peer reviewed \| Published
Community guidelines for GPCR ligand bias: IUPHAR review 32 Kolb, P; Kenakin, T; Alexander, S; Bermudez, M; Bohn, L; Breinholt; C; Bouvier, M; Hill, S; Kostenis, E; Martemyanov, K; Neubig, R; Onaran, O; Rajagopal, S; Roth, B; Selent, J; Shukla, A; Sommer, M; Gloriam D (2022) In: British Journal of Pharmacology, 179(14), 3651-3674. doi:10.1111/bph.15811 Review article (journal) \| Peer reviewed \| Published
Allosteric coupling and biased agonism in G protein‐coupled receptors Bock, A; Bermudez, M (2021) In: The FEBS Journal, 288, 2513-2528. doi:10.1111/febs.15783 Review article (journal) \| Peer reviewed \| Published
Antinociceptive Efficacy of the µ-Opioid/Nociceptin Peptide-Based Hybrid KGNOP1 in Inflammatory Pain without Rewarding Effects in Mice: An Experimental Assessment and Molecular Docking Dumitrascuta M, Bermudez M, Trovato O, Neve JD, Ballet S, Wolber G, Spetea M (2021) In: Molecules, 26, 3267-3267. doi:10.3390/molecules26113267 Research article (journal) \| Peer reviewed \| Published
Structure‐based identification of dual ligands at the A2AR and PDE10A with anti‐proliferative effects in lung cancer cell‐lines Kalash, L; Winfield, I; Safitri, D; Bermudez, M; Carvalho, S; Glen, R; Ladds, G; Bender, A (2021) In: Journal of Cheminformatics, 13(1), 17 (2021). doi:10.1186/s13321-021-00492-5 Research article (journal) \| Peer reviewed \| Published
Biological Characterization, Mechanistic Investigation and Structure‐Activity Relationships of Chemically Stable TLR2 Antagonists Bermudez M, Grabowski M, Murgueitio MS, Tiemann M, Varga P, Rudolf T, Wolber G, Weindl G, Rademann J (2020) In: ChemMedChem, 15, 1364-1371. doi:10.1002/cmdc.202000060 Research article (journal) \| Peer reviewed \| Published
Ligand-Specific Allosteric Coupling Controls G-Protein-Coupled Receptor Signaling Holze J, Bermudez M, Pfeil EM, Kauk M, Bödefeld T, Irmen M, Matera C, Dallanoce C, Amici MD, Holzgrabe U, König GM, Tränkle C, Wolber G, Schrage R, Mohr K, Hoffmann C, Kostenis E, Bock A (2020) In: ACS Pharmacology & Translational Science, 3(5), 859-867. doi:10.1021/acsptsci.0c00069 Research article (journal) \| Peer reviewed \| Published
Mechanistic Understanding of Peptide Analogues, DALDA, [Dmt1]DALDA, and KGOP01, Binding to the Mu Opioid Receptor Dumitrascuta M, Bermudez M, Ballet S, Wolber G, Spetea M (2020) In: Molecules, 25, 2087. doi:10.3390/molecules25092087 Research article (journal) \| Peer reviewed \| Published

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